GABA Receptor
GABA receptors are a class of receptors that respond to the neurotransmitter gamma-aminobutyric acid (GABA), the chief inhibitory compound in the mature vertebrate central nervous system. GABA receptors influence cognition by coordinating with glutamatergic processes. There are two classes of GABA receptors: GABAA and GABAB. GABAA receptors are ligand-gated ion channels; whereas GABAB receptors are G protein-coupled receptors, also called metabotropic receptors. A subclass of ionotropic GABA receptors, insensitive to typical allosteric modulators of GABAA receptor channels such as benzodiazepines and barbiturates, designated GABAС receptor.
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2-Hydroxysaclofen是选择性 GABAB 拮抗剂，比saclofen活性更强。。
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17-PA是Neurosteroid activation的拮抗剂，direct gating of GABAA。
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(S)-SNAP 5114是GABA uptake inhibitor（摄取抑制剂）。
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(RS)-Baclofen是选择性 GABAB 激动剂。
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(±)-Nipecotic acid是GABA uptake inhibitor（摄取抑制剂）。
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2-Hydroxysaclofen是选择性 GABAB 拮抗剂，比saclofen活性更强。。
More
-
17-PA是Neurosteroid activation的拮抗剂，direct gating of GABAA。
More
-
(S)-SNAP 5114是GABA uptake inhibitor（摄取抑制剂）。
More
-
(RS)-Baclofen是选择性 GABAB 激动剂。
More
-
(±)-Nipecotic acid是GABA uptake inhibitor（摄取抑制剂）。
More
